16-02-2014, 07:50 PM
An androgen antagonist (anti-androgen) can broadly be defined as any compound that has the biological effect of blocking or suppressing the action of male sex hormones such as testosterone within the human body. DHT blocks the conversion of aromatase (bad for breast growth).
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Reishi-reishi mushrooms significantly reduced levels of 5-alpha reductase, preventing conversion of testosterone into the more potent DHT. High levels of DHT are a risk factor for conditions such as benign prostatatic hypertrophy (BPH), acne, and baldness.
White Peony--Estrogenic, blocks 5ar and pro-aromatase - Strong.
A compound found in white peony inhibits the production of testosterone and promotes the activity of aromatase, which converts testosterone into estrogen.
Spearmint-anti-androgenic properties reduce the level of free testosterone in the blood, while leaving total testosterone and DHEAS unaffected.
Green Tea Epigallocatechin-Green tea (camellia)-Reduce's the conversion of free testosterone into DHT and also raises SHBG (sex-hormone-binding-globulin).
Pygeum-include phytosterols that inhibit the production of dht. Pygeum also reduce's prolacting levels and block the accumulation of cholesterol in the prostate. Prolactin increase's the uptake of testosterone by the prostate. Pygeum reduces the levels of DHT in the blood and reduces the number of sites where the dht can attach.
Saw palmetto-Saw palmetto-Beta-sitosterol is a natural alpha-adrenergic receptor blocker. Prevents DHT from accumulating in prostate tissue that would otherwise cause excessive cell growth and inflammation. The plant steroids in saw palmetto also act on progesterone receptors, an action that causes a reduction in estrogen levels.
DIM is Diindolylmethane-It is an anti carcinogen and also improves estrogen metabolism. Plant-derived 3,3′-Diindolylmethane Is a Strong Androgen Antagonist in Human Prostate Cancer Cells* DIM is remarkably similar in conformational geometry and surface charge distribution to an established synthetic AR antagonist, Taken with estrogen agonist, activities of DIM are seen as an hormone disrupter. DIM is the first example of a pure androgen receptor antagonist from plants.
Nettle Root- should be in the conversation
Nettle Root--Binds to SHBG (hormone that binds to excess hormones by decreasing hormone levels), and decreases 5ar and aromatase. Taking this tends to increase estrogen and testosterone. Would need to be taken with a pro-aromatase, and maybe estrogen.
Nettle root can interfere with or block a number these hormone-related chemical processes in the body that are implicated in the development of BPH. In clinical research, nettle has demonstrated the ability to stop the conversion of testosterone to dihydrotestosterone (by inhibiting aromatase, an enzyme required for the conversion), as well as to directly bind to SHBG itself - thereby preventing SHBG from binding to other hormones. Other research also reveals that nettles can prevent SHBG that has already bound to a hormone from attaching to the receptor sites on the prostate, as well as to decrease the production of estrogens (estradiol and estrone) by inhibiting an enzyme required for their production. The effect of nettle root on dihydrotestosterone (DHT) levels has also made it a treatment for hair loss, as male pattern balding has often been linked to an excess of DHT, as has hair loss in women too.
Chinese Skullcap should be in the conversation too-
Chinese Skullcap Inhibits the 5alpha-reductase enzyme-
Baicalein has been shown to inhibit the 5alpha-reductase enzyme, which converts testosterone to dihydrotestosterone (DHT). DHT is strongly associated with the development of prostate enlargement (benign prostatic hyperplasia) and prostate cancer. As such, baicalein is reported to be potentially useful for the prevention and/or treatment of androgen-dependent (testosterone-driven) disorders, including prostate enlargement and prostate cancer.
Licorice needs to be in the list
Use with extreme caution
Licorice (Glycyrrhiza glabra)-Anti-androgenic and activates alpha and beta estrogen receptors and blocks 5-ar - Strong, but take in moderation!
Licorice is a flavorful substance that has been used in food and medicinal remedies for thousands of years. It is also known as “sweet root,” licorice root contains a compound that is about 50 times sweeter than sugar. It has been used in both Eastern and Western medicine to treat a variety of illnesses ranging from the common cold to liver disease. Licorice affects the endocrine system because it contains isoflavones (phytoestrogens), which are chemicals found in plants that may mimic the effects of estrogen and relieve menopausal symptoms and menstrual disorders. Licorice may also reduce testosterone levels, which can contribute to hirsutism in women.
A small clinical trial published in 2004 by Armanini and colleagues found that licorice root significantly decreases testosterone levels in healthy female volunteers. Women taking daily licorice root experienced a drop in total testosterone levels after 1 month and testosterone levels returned to normal after discontinuation. It is unclear as to whether licorice root affects free testosterone levels. The endocrine effect is thought to be due to phytoestrogens and other chemicals found in licorice root, including the steroid glycyrrhizin and glycyrrhetic acid, which also have a weak anti-androgen effect
http://www.breastnexus.com/showthread.php?tid=5250
More about licorice-FOR REFERENCE (please add on as necessary)
I'm not sure how you would take LR at night before sleeping as it was suggested.
-Licorice root is the only herb that balances estrogen, stimulates prolactin, and blocks testosterone all at the same time. Licorice contains numerous phytoestrogenic compounds such as glabridin, glaberine, and 3-hydroxyglabrol.
-Beneficial for hypoglycemia, bronchitis, colitis, diverticulosis, gastritis, stress, colds, nausea, and inflammation. Cleanses the colon, promotes adrenal gland function, decreases muscle or skeletal spasms, and increases the fluidity of mucus from the lungs and bronchial tubes. Has estrogen-like hormone effects; changes the voice. Studies show licorice root stimulates the production of interferon. Warning: Do not use if you have high blood pressure."
-Researchers are currently excited about the diverse healing properties of licorice, from its anti-inflammatory abilities to its capacity to soothe stomach upset and control coughs. Even the National Cancer Institute has investigated the medicinal benefits of licorice.
-Lessen symptoms of chronic fatigue syndrome and fibromyalgia. By enhancing cortisol activity, glycyrrhizin helps to increase energy, ease stress, and reduce the symptoms of ailments sensitive to cortisol levels, such as chronic fatigue syndrome and fibromylagia. In the 1800s, licorice extract was a common remedy for a type of persistent fatigue known as neurasthenia, the condition now known as chronic fatigue syndrome.
-Soothe skin irritations such as eczema and shingles. Licorice cream applied directly to irritated skin can help to reduce inflammation and relieve such symptoms as itching and burning. It also boosts the effectiveness of cortisone creams.
-For most disorders: Take 200 mg standardized extract in pill form three times a day, or 20 to 45 drops, three times a day, of a 1:5 tincture. (The 1:5 tincture represents one part herb is soaked in five parts liquid
-Don't use licorice candy in place of supplements. Most red or black licorice candy sold in the United States contains anise oil as a flavoring rather than licorice. Candy made in Europe may contain licorice, but the quantities are not standardized.
-Licorice can raise blood pressure--a function of glycyrrhizin's action on the adrenal glands--so avoid taking more than the recommended dosage. If you take licorice for more than four weeks, have your blood pressure checked. (Stop taking the herb at the first sign of high blood pressure; this side effect is reversible.)
-At high doses taken over long periods of time, licorice can result in excessive salt loss from the blood, heart irregularities, and other serious health problems. Symptoms of this type of overdose may include headache, swelling, stiffness, shortness of breath, upper abdominal pain, and lethargy, among others.
-Side effects should disappear very shortly after stopping licorice. If not, see a doctor at once.
Sources:
http://www.breastnexus.com/showthread.php?tid=5250
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3693613/
http://endometabol.com/?page=article&article_id=3644
http://www.meschinohealth.com/ArticleDir..._Treatment
Abstracts-See frequently used supplements
____________________________________________________________________
Reishi-reishi mushrooms significantly reduced levels of 5-alpha reductase, preventing conversion of testosterone into the more potent DHT. High levels of DHT are a risk factor for conditions such as benign prostatatic hypertrophy (BPH), acne, and baldness.
White Peony--Estrogenic, blocks 5ar and pro-aromatase - Strong.
A compound found in white peony inhibits the production of testosterone and promotes the activity of aromatase, which converts testosterone into estrogen.
Spearmint-anti-androgenic properties reduce the level of free testosterone in the blood, while leaving total testosterone and DHEAS unaffected.
Green Tea Epigallocatechin-Green tea (camellia)-Reduce's the conversion of free testosterone into DHT and also raises SHBG (sex-hormone-binding-globulin).
Pygeum-include phytosterols that inhibit the production of dht. Pygeum also reduce's prolacting levels and block the accumulation of cholesterol in the prostate. Prolactin increase's the uptake of testosterone by the prostate. Pygeum reduces the levels of DHT in the blood and reduces the number of sites where the dht can attach.
Saw palmetto-Saw palmetto-Beta-sitosterol is a natural alpha-adrenergic receptor blocker. Prevents DHT from accumulating in prostate tissue that would otherwise cause excessive cell growth and inflammation. The plant steroids in saw palmetto also act on progesterone receptors, an action that causes a reduction in estrogen levels.
DIM is Diindolylmethane-It is an anti carcinogen and also improves estrogen metabolism. Plant-derived 3,3′-Diindolylmethane Is a Strong Androgen Antagonist in Human Prostate Cancer Cells* DIM is remarkably similar in conformational geometry and surface charge distribution to an established synthetic AR antagonist, Taken with estrogen agonist, activities of DIM are seen as an hormone disrupter. DIM is the first example of a pure androgen receptor antagonist from plants.
Nettle Root- should be in the conversation
Nettle Root--Binds to SHBG (hormone that binds to excess hormones by decreasing hormone levels), and decreases 5ar and aromatase. Taking this tends to increase estrogen and testosterone. Would need to be taken with a pro-aromatase, and maybe estrogen.
Nettle root can interfere with or block a number these hormone-related chemical processes in the body that are implicated in the development of BPH. In clinical research, nettle has demonstrated the ability to stop the conversion of testosterone to dihydrotestosterone (by inhibiting aromatase, an enzyme required for the conversion), as well as to directly bind to SHBG itself - thereby preventing SHBG from binding to other hormones. Other research also reveals that nettles can prevent SHBG that has already bound to a hormone from attaching to the receptor sites on the prostate, as well as to decrease the production of estrogens (estradiol and estrone) by inhibiting an enzyme required for their production. The effect of nettle root on dihydrotestosterone (DHT) levels has also made it a treatment for hair loss, as male pattern balding has often been linked to an excess of DHT, as has hair loss in women too.
Chinese Skullcap should be in the conversation too-
Chinese Skullcap Inhibits the 5alpha-reductase enzyme-
Baicalein has been shown to inhibit the 5alpha-reductase enzyme, which converts testosterone to dihydrotestosterone (DHT). DHT is strongly associated with the development of prostate enlargement (benign prostatic hyperplasia) and prostate cancer. As such, baicalein is reported to be potentially useful for the prevention and/or treatment of androgen-dependent (testosterone-driven) disorders, including prostate enlargement and prostate cancer.
Licorice needs to be in the list
Use with extreme caution
Licorice (Glycyrrhiza glabra)-Anti-androgenic and activates alpha and beta estrogen receptors and blocks 5-ar - Strong, but take in moderation!
Licorice is a flavorful substance that has been used in food and medicinal remedies for thousands of years. It is also known as “sweet root,” licorice root contains a compound that is about 50 times sweeter than sugar. It has been used in both Eastern and Western medicine to treat a variety of illnesses ranging from the common cold to liver disease. Licorice affects the endocrine system because it contains isoflavones (phytoestrogens), which are chemicals found in plants that may mimic the effects of estrogen and relieve menopausal symptoms and menstrual disorders. Licorice may also reduce testosterone levels, which can contribute to hirsutism in women.
A small clinical trial published in 2004 by Armanini and colleagues found that licorice root significantly decreases testosterone levels in healthy female volunteers. Women taking daily licorice root experienced a drop in total testosterone levels after 1 month and testosterone levels returned to normal after discontinuation. It is unclear as to whether licorice root affects free testosterone levels. The endocrine effect is thought to be due to phytoestrogens and other chemicals found in licorice root, including the steroid glycyrrhizin and glycyrrhetic acid, which also have a weak anti-androgen effect
http://www.breastnexus.com/showthread.php?tid=5250
More about licorice-FOR REFERENCE (please add on as necessary)
I'm not sure how you would take LR at night before sleeping as it was suggested.
-Licorice root is the only herb that balances estrogen, stimulates prolactin, and blocks testosterone all at the same time. Licorice contains numerous phytoestrogenic compounds such as glabridin, glaberine, and 3-hydroxyglabrol.
-Beneficial for hypoglycemia, bronchitis, colitis, diverticulosis, gastritis, stress, colds, nausea, and inflammation. Cleanses the colon, promotes adrenal gland function, decreases muscle or skeletal spasms, and increases the fluidity of mucus from the lungs and bronchial tubes. Has estrogen-like hormone effects; changes the voice. Studies show licorice root stimulates the production of interferon. Warning: Do not use if you have high blood pressure."
-Researchers are currently excited about the diverse healing properties of licorice, from its anti-inflammatory abilities to its capacity to soothe stomach upset and control coughs. Even the National Cancer Institute has investigated the medicinal benefits of licorice.
-Lessen symptoms of chronic fatigue syndrome and fibromyalgia. By enhancing cortisol activity, glycyrrhizin helps to increase energy, ease stress, and reduce the symptoms of ailments sensitive to cortisol levels, such as chronic fatigue syndrome and fibromylagia. In the 1800s, licorice extract was a common remedy for a type of persistent fatigue known as neurasthenia, the condition now known as chronic fatigue syndrome.
-Soothe skin irritations such as eczema and shingles. Licorice cream applied directly to irritated skin can help to reduce inflammation and relieve such symptoms as itching and burning. It also boosts the effectiveness of cortisone creams.
-For most disorders: Take 200 mg standardized extract in pill form three times a day, or 20 to 45 drops, three times a day, of a 1:5 tincture. (The 1:5 tincture represents one part herb is soaked in five parts liquid
-Don't use licorice candy in place of supplements. Most red or black licorice candy sold in the United States contains anise oil as a flavoring rather than licorice. Candy made in Europe may contain licorice, but the quantities are not standardized.
-Licorice can raise blood pressure--a function of glycyrrhizin's action on the adrenal glands--so avoid taking more than the recommended dosage. If you take licorice for more than four weeks, have your blood pressure checked. (Stop taking the herb at the first sign of high blood pressure; this side effect is reversible.)
-At high doses taken over long periods of time, licorice can result in excessive salt loss from the blood, heart irregularities, and other serious health problems. Symptoms of this type of overdose may include headache, swelling, stiffness, shortness of breath, upper abdominal pain, and lethargy, among others.
-Side effects should disappear very shortly after stopping licorice. If not, see a doctor at once.
Sources:
http://www.breastnexus.com/showthread.php?tid=5250
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3693613/
http://endometabol.com/?page=article&article_id=3644
http://www.meschinohealth.com/ArticleDir..._Treatment
Abstracts-See frequently used supplements